Preclinical Stage

Drug discovery, redefined by computation.

Axia Discovery combines physics-based molecular simulation, generative AI, and multi-omics data to identify and validate novel drug candidates — faster, and with greater precision than conventional approaches.

De Novo
Generative peptide design
In Silico
Designed before synthesis
10
Patent-pending programs
The Axia Platform

End-to-end computational drug discovery

From target to candidate, our integrated platform compresses timelines while elevating the quality of every decision.

Target Identification

Genomics · Proteomics

Multi-omics and network-biology integration to prioritize disease-relevant receptor targets with high therapeutic confidence.

De Novo Design

Generative AI · De Novo

Generative AI designs novel cyclic-peptide binders from scratch against a chosen target — ownable compositions of matter, not library hits.

Physics-Based Simulation

Physics-Based

Physics-based molecular simulation models how candidates bind and behave, prioritizing the most selective, highest-quality designs before synthesis.

Selectivity by Design

Selectivity

Candidates are engineered to discriminate the intended target from its closest receptor relatives — selectivity built in from the first design.

Developability

PK/PD · Safety

Computational assessment of developability, PK, and safety liabilities early in the campaign — surfacing risk before the wet lab.

Lead Refinement

Iterative Design

Iterative design-and-assess cycles refine each candidate toward its target product profile.

Pipeline

Ten patent-pending programs

Led by oncology radioligand therapy, with CNS, cardiometabolic, and renal programs — de novo-designed cyclic peptides. 11 U.S. provisional patent applications filed 2026.

Full pipeline →
Target ID
Design
Hit-to-Lead
Lead Opt.
Preclinical
Oncology · Radioligand Therapy
AX-RLT-001patent pending
Castration-resistant prostate cancer (beyond current radioligand therapy)
Undisclosed
Preclinical
AX-RLT-002patent pending
Prostate / ER+ breast cancer
Undisclosed
Preclinical
AX-RLT-003patent pending
Endometrial carcinoma
Undisclosed
Preclinical
Oncology · Composition IP (non-radiation)
AX-PDC-001patent pending
Multiple myeloma
Undisclosed
Preclinical
AX-PDC-002patent pending
Solid tumors
Undisclosed
Preclinical
CNS / Neuropsychiatry
AX-CP-001patent pending
Neurological disorders
Undisclosed
Preclinical
AX-CP-002patent pending
Depression / anxiety · DEE / obesity
Undisclosed
Preclinical
Cardiometabolic
AX-CP-003patent pending
Heart failure / PAH / cardiometabolic
Undisclosed
Preclinical
AX-CP-004patent pending
Obesity / metabolic
Undisclosed
Preclinical
Renal
AX-CP-005patent pending
Secondary hyperparathyroidism (CKD-MBD)
Undisclosed
Preclinical

Preclinical · in-silico-designed, wet-lab validation underway · patent pending · PCT international filings anticipated · Pipeline subject to change

Scientific Foundation

Rigorous methodology, measurable outcomes

Physics-based simulation and generative AI, applied with discipline at every step — novel candidates designed in silico, with wet-lab validation underway.

De Novo
Generative peptide design
Designed from scratch, not library-screened
In Silico
Designed before synthesis
Wet-lab validation underway
Physics + AI
Hybrid platform
Physics-based simulation + generative AI
10
Patent-pending programs
11 U.S. provisionals filed 2026
Partner with Axia

Ready to accelerate your drug discovery program?

Whether you're seeking a computational co-development partner, licensing opportunities, or looking to advance a difficult target — let's talk.