In Silico Pipeline

Computational Drug Discovery in Action

Our preclinical pipeline combines peptide chemistry with cutting-edge in-silico methods. All programs are built on validated computational workflows, from target identification through lead optimization.

AXD-001

Lead Program

Oncology — Solid Tumors

Target

Undisclosed peptide target

Lead peptide optimization underway. Target validation complete. Next phase: structure-activity relationship refinement.

DEVELOPMENT STAGE

Hit-to-Lead

AXD-002

Neurodegeneration

Target

Amyloidogenic peptide modulator

Computational screening against target database. Identifying hit series with predicted ADMET properties. Validation pending.

DEVELOPMENT STAGE

Virtual Screening

AXD-003

Inflammatory Disease

Target

Undisclosed peptide target

Target characterization in progress. Bioinformatic analysis complete. Virtual screening pipeline preparation underway.

DEVELOPMENT STAGE

Target Validation

How Our Pipeline Works

Target Identification & Validation

We use computational methods to identify and validate novel peptide targets based on disease biology, biomarker data, and literature mining.

Virtual Screening

Our platform screens billions of peptide-like molecules against validated targets using structure-based and ligand-based computational methods.

Hit-to-Lead Optimization

Computational design of improved analogs with enhanced potency, selectivity, and ADMET properties through iterative de novo design.

Lead Optimization

Final refinement for preclinical candidate selection, including metabolic stability, off-target effects, and in vivo performance prediction.

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